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SR-4835

Glpbio
Catalog No:GC39175-10mM (in 1mL DMSO) CAS No.:2387704-62-1 MDLNo: Brand:Glpbio purity: 特性: Purpose:SR-4835 是有效,高选择性和 ATP 竞争性的 CDK12/CDK13 双重抑制剂 (CDK12:IC50=99 nM,Kd=98 nM;CDK13:Kd=4.9 nM)。SR-4835 与破坏 DNA 的化学疗法和 PARP 抑制剂协同作用,并引起三阴性乳腺癌 (TNBC) 细胞凋亡。DMSO: 5 mg/mL (10.01 mM; ultrasonic and warming and heat to 60°C)
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